Basic Peptide Information

DICL ID
DICL_Pep_07074
Ion Channel
Sodium channel protein type 3 subunit alpha
Peptide Function
Blocker
Gene Name
Scn3a

Activity Data (nM)

IC50
8000 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
CCNCSSKWCRDHSRCC
Peptide UniProt Accession
UniParc
UPI0000603521
Peptide Synonyms/Alias
[mu-Conotoxin K IIIA; UNII-390H5GUO40; CHEMBL2402969; 390H5GUO40; 884469-67-4; Ccncsskwcrdhsrcc-NH2 cyclic (1->9);(2->15);(4->16); L-Cysteinamide; L-cysteinyl-L-cysteinyl-L-asparaginyl-L-cysteinyl-L-seryl-L-seryl-L-lysyl-L-tryptophyl-L-cysteinyl-L-arginyl-L-alpha-aspartyl-L-histidyl-L-seryl-L-arginyl-L-cysteinyl-; cyclic (1->9);(2->15);(4->16)-tris(disulfide); mu-Conotoxin KIIIA; BDBM50492340; DA-68915]
Peptide Species
Conus kinoshitai
Peptide Name
Mu-conotoxin KIIIB
CAS Number
884469-67-4

Experimental Conditions

pH
pH 7.3
Holding Potential (mV)
−80 mV
Temperature
21−24 °C
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available